Cart
sales@molnova.com
ICI 174,864
CAS No. 89352-67-0
ICI 174,864( —— )
Catalog No. M30662 CAS No. 89352-67-0
Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 387 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
Biological Information
-
Product NameICI 174,864
-
NoteResearch use only, not for human use.
-
Brief DescriptionSelective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
-
DescriptionSelective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayEndocrinology/Hormones
-
TargetOpioid Receptor
-
Recptor——
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number89352-67-0
-
Formula Weight691.87
-
Molecular FormulaC38H53N5O7
-
Purity>98% (HPLC)
-
SolubilityDMSO:69.19 mg/mL;water:1 mg/ml
-
SMILESCC(C)C[C@H](NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)C(C)(C)NC(=O)C(C)(C)NC(=O)[C@H](CC1=CC=C(O)C=C1)N(CC=C)CC=C)C(O)=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Cohen et al (1996) Opioid agonist activity of ICI 174864 and its carboxypeptidase degradation product, LY281217. J.Pharmacol.Exp.Ther. 238 769 PMID:
molnova catalog
related products
-
Trimebutine
Trimebutine is a drug with antimuscarinic and weak mu opioid agonist effects.
-
BTRX-335140
BTRX-335140 is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively.
-
Adrenorphin(3TFA)
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
